SCHEMBL5068834

SCHEMBL5068834

O=C(O)N(Cc1cccc(CC(Cl)=CCl)c1)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGER Q15109 3/20 0.41
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
OPRM1 P35372 2/20 0.41
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
CTSD P07339 1/20 0.40
TACR1 P25103 2/20 0.39
DCUN1D1 Q96GG9 2/20 0.39
ALDH1A1 P00352 1/20 0.39
THRB P10828 1/20 0.39
MTNR1A P48039 1/20 0.39
KCNH2 Q12809 1/20 0.39
PTGES O14684 1/20 0.38
UBE2M P61081 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370759 0.78 AGER (0.55) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL5913502 0.76 HSD11B1 (0.47) AGERCHRM2CHRM3OPRM1SLC6A2
SCHEMBL3373057 0.74 AGER (0.58) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL736913 0.72 AGER (0.50) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL736914 0.72 AGER (0.50) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL18586065 0.72 HDAC8 (0.43) AGERCHRM2CHRM3OPRM1SLC6A2
SCHEMBL17506917 0.72 MC4R (0.49) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL1700010 0.72 MC4R (0.49) AGERCHRM2CHRM3OPRM1CTSD
SCHEMBL1069848 0.72 SLC6A2 (0.42) AGERCHRM2CHRM3OPRM1SLC6A2
SCHEMBL77425 0.71 MC4R (0.54) AGERCHRM2CHRM3OPRM1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910272-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2008-04-16 EP disclosed
WO-2007009250-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-01-25 WO disclosed