SCHEMBL5069502

SCHEMBL5069502

CCCc1ccnc(OC)c1OC

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HMGCR P04035 1/20 0.34
DHFR P00374 2/20 0.34
MTNR1A P48039 2/20 0.33
SREBF2 Q12772 2/20 0.33
ACSS2 Q9NR19 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NOS2 P35228 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
MAOA P21397 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
RPS6KA5 O75582 1/20 0.32
MTNR1B P49286 1/20 0.32
SLC13A5 Q86YT5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5072115 0.81 ACSS2 (0.34) ALDH1A1MAPTMTNR1AACSS2MAOA
SCHEMBL19330160 0.79 MEN1 (0.39) ALDH1A1MAPTMTNR1AACSS2SMN1; SMN2
SCHEMBL19330347 0.79 HPGD (0.34) ALDH1A1MAPTMTNR1AACSS2HPGD
SCHEMBL30701188 0.79 MEN1 (0.39) ALDH1A1MAPTMTNR1AACSS2SMN1; SMN2
SCHEMBL28118987 0.78 KDM4E (0.39) ALDH1A1MAPTMTNR1AMTNR1B
SCHEMBL12093550 0.76 SLC13A5 (0.51) ADRA2AADRA2BADRA2CMAOASLC13A5
SCHEMBL28301401 0.75 PPARA (0.43) MTNR1AMTNR1BSLC13A5
SCHEMBL6645213 0.74 HSD17B10 (0.41) ALDH1A1MAPTMTNR1AHPGDSLC13A5
SCHEMBL5072695 0.74 CYP3A4 (0.42) ALDH1A1MAPTMTNR1AACSS2SMN1; SMN2
SCHEMBL24344519 0.72 AURKA (0.38) MTNR1AHPGDSMN1; SMN2NOS2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007386-A2 CAMPTOTHECIN-ANALOG WITH A NOVEL, FLIPPED LACTONE-STABLE, E-RING AND METHODS FOR MAKING AND USING SAME BIONUMERIK PHARMACEUTICALS, INC. (US) 2008-12-31 EP disclosed
WO-2007123995-A2 CAMPTOTHECIN-ANALOG WITH A NOVEL, “FLIPPED” LACTONE-STABLE, E-RING AND METHODS FOR MAKING AND USING SAME BIONUMERIK PHARMACEUTICALS, INC. (US) 2007-11-01 WO disclosed
EP-0035893-A2 Herbicidal benzene- and pyridine-sulfonamide derivatives E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-09-16 EP disclosed