SCHEMBL5072287

SCHEMBL5072287

COCCCc1ncc(Cl)c(CN(C(=O)C(CNC(=O)O)Cc2ccc(OCCOc3c(Cl)cc(C)cc3Cl)cc2)C2CC2)c1O

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.62
CYP3A4 P08684 7/20 0.62
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5071357 0.89 REN (0.60) RENCYP3A4KCNH2
SCHEMBL5072283 0.87 REN (0.52) RENCYP3A4
SCHEMBL4349864 0.87 REN (0.75) RENCYP3A4
SCHEMBL5072291 0.85 REN (0.65) RENCYP3A4
SCHEMBL4351920 0.83 REN (0.58) RENCYP3A4
SCHEMBL661618 0.83 REN (0.76) RENCYP3A4
SCHEMBL4354028 0.83 REN (0.56) RENCYP3A4
SCHEMBL4347867 0.83 CYP3A4 (0.68) RENCYP3A4KCNH2
SCHEMBL4349317 0.83 CYP3A4 (0.66) RENCYP3A4KCNH2
SCHEMBL664368 0.82 CYP3A4 (0.71) RENCYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910272-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2008-04-16 EP disclosed
WO-2007009250-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-01-25 WO disclosed