SCHEMBL5073180

SCHEMBL5073180

O=C(O)c1cn2c3c(sc2n1)COCC3

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PTPRC P08575 1/20 0.36
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
PTPRB P23467 1/20 0.36
PTPRE P23469 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
FABP4 P15090 12/20 0.35
FABP5 Q01469 12/20 0.35
HDAC6 Q9UBN7 1/20 0.33
PDK1 Q15118 1/20 0.32
GAA P10253 1/20 0.32
NFKB1 P19838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3588423 0.81 GAA (0.43) NPC1ALDH1A1MAPTRAB9AKMT2A
SCHEMBL17620987 0.80 ALDH1A1 (0.56) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL17620969 0.78 ALDH1A1 (0.55) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL3593173 0.78 NPC1 (0.34) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL13455807 0.75 HDAC6 (0.36) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL17621010 0.73 FABP4 (0.39) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL3212977 0.71 LIMK1 (0.35) PTPRCPTPN2PTPN1PTPRBPTPRE
SCHEMBL17620989 0.70 FABP4 (0.38) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL17620984 0.70 MAPT (0.40) NPC1ALDH1A1TP53MAPTRAB9A
SCHEMBL3600663 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909786-A2 TRICYCLIC 6-ALKYLIDENE-PENEM ß-LACTAMASE INHIBITORS AND ß-LACTAM ANTIBIOTIC COMBINATION: A BROAD SPECTRUM ANTIBIOTIC Wyeth a Corporation of the State of Delaware (US) 2008-04-16 EP disclosed
WO-2007027323-A2 TRICYCLIC 6-ALKYLIDENE-PENEM β-LACTAMASE INHIBITORS AND β-LACTAM ANTIBIOTIC COMBINATION: A BROAD SPECTRUM ANTIBIOTIC WYETH (US) 2007-03-08 WO disclosed