SCHEMBL5074208

SCHEMBL5074208

[CH2]CCCCCCCCCCCCCCSCCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.53
CYP2D6 P10635 3/20 0.53
CYP2C19 P33261 3/20 0.53
CA2 P00918 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CES1 P23141 2/20 0.41
SIGMAR1 Q99720 6/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NOS1 P29475 1/20 0.38
MAOA P21397 2/20 0.38
NPC1 O15118 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5975773 0.98 CYP1A2 (0.55) CYP1A2CYP2D6CYP2C19CA2CYP3A4
SCHEMBL5979562 0.92 CA2 (0.51) CYP1A2CYP2D6CYP2C19CA2SIGMAR1
SCHEMBL2730659 0.92 CYP1A2 (0.57) CYP1A2CYP2D6CYP2C19CA2CYP3A4
SCHEMBL5974863 0.86 CA2 (0.53) CYP1A2CYP2D6CYP2C19CA2SIGMAR1
Ammonia Solution, Strong SCHEMBL23014996 0.85 SIGMAR1 (0.46) CYP1A2CYP2D6CYP2C19CA2SIGMAR1
SCHEMBL5073228 0.84 CYP2C19 (0.48) CYP1A2CYP2D6CYP2C19CA2CYP3A4
SCHEMBL539499 0.84 CYP2C19 (0.48) CYP1A2CYP2D6CYP2C19CA2CYP3A4
SCHEMBL8082718 0.83 SIGMAR1 (0.56) CYP1A2CYP2D6CYP2C19CA2SIGMAR1
SCHEMBL5975033 0.83 CYP1A2 (0.61) CYP1A2CYP2D6CYP2C19CA2CYP3A4
SCHEMBL10963241 0.83 SIGMAR1 (0.56) CYP1A2CYP2D6CYP2C19CA2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697465-B1 POLYMER NANOCOMPOSITES AND METHODS FOR THEIR PREPARATION GEN ELECTRIC (US) 2008-02-13 EP disclosed
EP-1697465-A2 POLYMER NANOCOMPOSITES AND METHODS FOR THEIR PREPARATION GENERAL ELECTRIC COMPANY (US) 2006-09-06 EP disclosed
WO-2005061623-A2 POLYMER NANOCOMPOSITES AND METHODS FOR THEIR PREPARATION GENERAL ELECTRIC COMPANY (US) 2005-07-07 WO disclosed
US-20050137310-A1 Polymer nanocomposites and methods for their preparation CITIBANK, N.A., AS COLLATERAL AGENT 2005-06-23 US disclosed
US-5747560-A AMMONIUM SALTS ALLIEDSIGNAL INC. (US) 1998-05-05 US disclosed
EP-0598836-B1 MELT PROCESS FORMATION OF POLYMER NANOCOMPOSITE OF EXFOLIATED LAYERED MATERIAL ALLIED SIGNAL INC (US) 1997-10-15 EP disclosed
EP-0668888-A1 NANOCOMPOSITES OF GAMMA PHASE POLYMERS AlliedSignal Inc. (US) 1995-08-30 EP disclosed
US-5385776-A Polylactams ALLIEDSIGNAL INC. 1995-01-31 US disclosed
EP-0598836-A1 MELT PROCESS FORMATION OF POLYMER NANOCOMPOSITE OF EXFOLIATED LAYERED MATERIAL. ALLIED SIGNAL INC (US) 1994-06-01 EP disclosed
WO-1994011430-A1 NANOCOMPOSITES OF GAMMA PHASE POLYMERS ALLIED-SIGNAL INC. (US) 1994-05-26 WO disclosed
WO-1993004117-A1 MELT PROCESS FORMATION OF POLYMER NANOCOMPOSITE OF EXFOLIATED LAYERED MATERIAL ALLIED-SIGNAL INC. (US) 1993-03-04 WO disclosed
WO-1993004118-A1 MELT PROCESS FORMATION OF POLYMER NANOCOMPOSITE OF EXFOLIATED LAYERED MATERIAL ALLIED-SIGNAL INC. (US) 1993-03-04 WO disclosed