SCHEMBL5074377

SCHEMBL5074377

Cc1cc(C)c2cc(Oc3c(Br)cccc3Br)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
ALDH1A1 P00352 4/20 0.40
HSD17B10 Q99714 4/20 0.40
POLB P06746 4/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
KDM4E B2RXH2 3/20 0.40
HPGD P15428 3/20 0.40
NQO2 P16083 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
SLC2A1 P11166 1/20 0.38
RAD52 P43351 1/20 0.38
PTPN11 Q06124 1/20 0.38
LMNA P02545 2/20 0.37
TSHR P16473 2/20 0.37
BCHE P06276 2/20 0.37
ACHE P22303 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5073565 0.82 KDM4E (0.38) ALDH1A1HSD17B10POLBKDM4EHPGD
SCHEMBL3142092 0.79 KDM4E (0.46) CYP1A2ALDH1A1HSD17B10POLBKDM4E
SCHEMBL3135783 0.78 KDM4E (0.43) CYP1A2ALDH1A1HSD17B10POLBKDM4E
SCHEMBL3135791 0.78 KDM4E (0.43) CYP1A2ALDH1A1HSD17B10POLBKDM4E
SCHEMBL3140997 0.78 THRA (0.55) CYP1A2ALDH1A1HSD17B10POLBKDM4E
SCHEMBL8103092 0.75 POLB (0.66) CYP1A2ALDH1A1HSD17B10POLBKDM4E
SCHEMBL30048942 0.71 CYP1A2 (0.57) CYP1A2ALDH1A1POLBKDM4ELMNA
SCHEMBL15724648 0.71 CYP1A2 (0.57) CYP1A2ALDH1A1POLBKDM4ELMNA
SCHEMBL19983503 0.71 ALDH1A1 (0.67) CYP1A2ALDH1A1HSD17B10POLBCASP1
SCHEMBL1161098 0.69 POLB (0.60) ALDH1A1HSD17B10POLBKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899309-A1 HETEROCYCLIC COMPOUNDS AS AGONISTS FOR THE THYROID RECEPTOR KARO BIO AB (SE) 2008-03-19 EP disclosed
WO-2007003419-A1 HETEROCYCLIC COMPOUNDS AS AGONISTS FOR THE THYROID RECEPTOR KARO BIO AB (SE) 2007-01-11 WO disclosed