SCHEMBL5074670

SCHEMBL5074670

CCC(=O)OC[C@H]1O[C@@H](n2ccc(=O)[nH]c2=O)[C@H](OC(=O)CC)[C@@H]1OC(=O)CC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HIF1A Q16665 1/20 0.48
SLC28A1 O00337 1/20 0.48
SLC28A2 O43868 1/20 0.48
SLC29A1 Q99808 1/20 0.48
SLC28A3 Q9HAS3 1/20 0.48
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.47
P2RY6 Q15077 7/20 0.46
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
P2RY2 P41231 9/20 0.46
P2RY12 Q9H244 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13901221 0.91 SLC28A1 (0.46) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL13901225 0.91 LMNA (0.46) LMNATHRBSMN1; SMN2HIF1ASLC28A1
SCHEMBL13901223 0.91 SLC28A1 (0.50) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL9556855 0.90 SLC28A1 (0.46) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL6222233 0.90 SLC28A1 (0.58) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL13901219 0.90 SLC28A1 (0.58) SLC28A1SLC28A2SLC29A1SLC28A3P2RY6
SCHEMBL5566835 0.89 CA12 (0.47) LMNATHRBSMN1; SMN2HIF1ASLC28A1
SCHEMBL13901227 0.88 LMNA (0.43) LMNATHRBSMN1; SMN2HIF1ASLC28A1
SCHEMBL9069522 0.87 CA12 (0.49) LMNATHRBSMN1; SMN2HIF1ASLC28A1
SCHEMBL24780787 0.87 LMNA (0.47) LMNATHRBSMN1; SMN2HIF1ASLC28A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7105498-B2 Acylated uridine and cytidine and uses thereof WELLSTAT THERAPEUTICS CORPORATION (US) 2006-09-12 US claimed
US-6274563-B1 ADMINISTERING AS ANTIDIABETIC AGENT PRO-NEURON, INC. 2001-08-14 US claimed
US-6258795-B1 Acylated uridine and cytidine and uses thereof PRO-NEURON, INC. 2001-07-10 US claimed
JP-2894610-B2 1999-05-24 JP claimed
US-5470838-A Method of delivering exogenous uridine or cytidine using acylated uridine or cytidine PRO-NEURON, INC. (US) 1995-11-28 US claimed
EP-0339075-B1 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF PRO-NEURON, INC. (US) 1993-08-18 EP claimed
EP-0339075-A4 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF. PRO NEURON INC (US) 1990-04-10 EP claimed
EP-0339075-A1 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF PRO-NEURON, INC. (US) 1989-11-02 EP claimed
WO-1989003837-A1 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF PRO-NEURON, INC. (US) 1989-05-05 WO claimed
EP-1778223-A4 METHODS AND COMPOSITIONS FOR REDUCING TOXICITY ASSOCIATED WITH LEFLUNOMIDE TREATMENT WILLIAMS JAMES W (US) 2008-03-05 EP disclosed
EP-1778223-A1 METHODS AND COMPOSITIONS FOR REDUCING TOXICITY ASSOCIATED WITH LEFLUNOMIDE TREATMENT Williams, James W. (US) 2007-05-02 EP disclosed
WO-2006014827-A1 METHODS AND COMPOSITIONS FOR REDUCING TOXICITY ASSOCIATED WITH LEFLUNOMIDE TREATMENT UNIV CHICAGO (US) 2006-02-09 WO disclosed
US-6316426-B1 NUCLEOSIDE DERIVATIVE FOR DIABETES, HEART DISEASE, CEREBROVASCULAR DISORDERS, PARKINSON'S DISEASE, INFANT RESPIRATORY DISTRESS SYNDROME AND FOR ENHANCEMENT OF PHOSPHOLIPID BIOSYNTHESIS PRO-NEURON, INC. 2001-11-13 US disclosed
US-6274563-B1 ADMINISTERING AS ANTIDIABETIC AGENT PRO-NEURON, INC. 2001-08-14 US disclosed
US-6258795-B1 Acylated uridine and cytidine and uses thereof PRO-NEURON, INC. 2001-07-10 US disclosed
US-5470838-A Method of delivering exogenous uridine or cytidine using acylated uridine or cytidine PRO-NEURON, INC. (US) 1995-11-28 US disclosed
EP-0339075-B1 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF PRO-NEURON, INC. (US) 1993-08-18 EP disclosed
EP-0339075-A1 ACYLATED URIDINE AND CYTIDINE AND USES THEREOF PRO-NEURON, INC. (US) 1989-11-02 EP disclosed