SCHEMBL5075615

SCHEMBL5075615

Cc1ccc(C(N)=O)c(C2CC2)c1Nc1ccc2c(c1)CC(C)(C)C2=O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.34
HDAC6 Q9UBN7 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSP90AA1 P07900 2/20 0.31
HSP90AB1 P08238 2/20 0.31
CSF1R P07333 1/20 0.31
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
CAMK1D Q8IU85 1/20 0.30
ESR1 P03372 2/20 0.30
ESR2 Q92731 2/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5285564 0.73 MAPK14 (0.38) MAPK14HDAC6
SCHEMBL3051840 0.72 TSHR (0.37) MAPK14ALDH1A1MAPT
SCHEMBL3054278 0.70 MAPK14 (0.59) MAPK14NPC1ALDH1A1MAPTRAB9A
SCHEMBL5076262 0.70 MAPK14 (0.40) MAPK14ALDH1A1
SCHEMBL5138721 0.70 MAPK14 (0.47) MAPK14NPC1ALDH1A1RAB9A
SCHEMBL3051914 0.69 MAPK14 (0.39) MAPK14
SCHEMBL3051000 0.69 MAPK14 (0.48) MAPK14NPC1ALDH1A1MAPTRAB9A
SCHEMBL3061264 0.69 MAPK14 (0.48) MAPK14NPC1MAPTSMN1; SMN2
SCHEMBL3048385 0.69 MAPK14 (0.65) MAPK14
SCHEMBL3056347 0.69 MAPK14 (0.43) MAPK14NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907358-A2 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS Palau Pharma, S.A. (ES) 2008-04-09 EP disclosed
WO-2007000340-A2 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO disclosed