SCHEMBL5078645

SCHEMBL5078645

CCc1ccc(OC(CCN(C)C)c2cccnc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.51
SLC6A2 P23975 2/20 0.51
SLC6A3 Q01959 1/20 0.51
HRH3 Q9Y5N1 2/20 0.49
ALDH1A1 P00352 2/20 0.48
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
CHRNA7 P36544 1/20 0.41
MAPT P10636 1/20 0.41
POLB P06746 1/20 0.39
SLC6A9 P48067 4/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP51A1 Q16850 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL2631 0.90 ALDH1A1 (0.48) SLC6A4SLC6A2SLC6A3HRH3ALDH1A1
Fumaric Acid SCHEMBL2633 0.90 ALDH1A1 (0.48) SLC6A4SLC6A2SLC6A3HRH3ALDH1A1
SCHEMBL11239618 0.74 SLC6A4 (0.68) SLC6A4SLC6A2HRH3SLC6A9
SCHEMBL2632 0.74 SLC6A2 (0.43) SLC6A4SLC6A2SLC6A3ALDH1A1MAPT
SCHEMBL5080333 0.73 CACNA2D1 (0.57) SLC6A4SLC6A2
Iodide SCHEMBL2607 0.72 CACNA2D1 (0.56) SLC6A4SLC6A2
SCHEMBL7158810 0.72 SLC6A4 (0.73) SLC6A4SLC6A2HRH3SLC6A9
SCHEMBL12620670 0.71 SLC6A4 (0.50) SLC6A4HRH3SLC6A9
SCHEMBL15809601 0.70 SLC6A4 (0.62) SLC6A4SLC6A2HRH3SLC6A9
Fumaric Acid SCHEMBL5313492 0.70 SLC6A2 (0.44) SLC6A4SLC6A2SLC6A3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008133884-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-11-06 WO disclosed