SCHEMBL5079780

SCHEMBL5079780

Cc1csc2sc(CN(C)C(=O)C=Cc3cnc(N)c(CN4CCOCC4)c3)c(C)c12

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 3/20 0.36
TBK1 Q9UHD2 3/20 0.36
KDM4E B2RXH2 3/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
RECQL P46063 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
CNR2 P34972 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5079778 1.00 IKBKE (0.36) IKBKETBK1KDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL1251887 0.99 IKBKE (0.36) IKBKETBK1KDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL1251890 0.99 IKBKE (0.36) IKBKETBK1KDM4EMAPTALDH1A1
SCHEMBL5079756 0.82 KDM4E (0.38) KDM4EMAPTSMN1; SMN2
SCHEMBL5079762 0.82 KDM4E (0.38) KDM4EMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL1253910 0.81 KDM4E (0.39) KDM4EMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL1253912 0.81 KDM4E (0.39) KDM4EMAPTSMN1; SMN2
SCHEMBL5079082 0.77 SMN1; SMN2 (0.39) KDM4EMAPTSMN1; SMN2
SCHEMBL726656 0.76 BMP1 (0.37)
SCHEMBL726657 0.76 BMP1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608377-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING INHIBITORS OF FAB I AND FURTHER ANTIBIOTICS AFFINIUM PHARM INC (CA) 2008-10-01 EP claimed