SCHEMBL5082011

SCHEMBL5082011

Nc1ccc(O)c(CCCl)c1CCCl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
ALOX15 P16050 4/20 0.35
HSD17B10 Q99714 4/20 0.35
HPGD P15428 2/20 0.35
ALOX12 P18054 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
HDAC3 O15379 1/20 0.35
IDO1 P14902 1/20 0.35
EP300 Q09472 1/20 0.35
KAT2B Q92831 1/20 0.35
KAT8 Q9H7Z6 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
GAA P10253 5/20 0.34
MAPT P10636 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 3/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133372 0.86 CYP3A4 (0.32) ALDH1A1ALOX15SMN1; SMN2CYP3A4TP53
Hydrochloric Acid SCHEMBL7517167 0.84 CYP3A4 (0.33) ALDH1A1ALOX15SMN1; SMN2MAPK1CYP3A4
SCHEMBL6573311 0.83 CNR1 (0.41) ALDH1A1ALOX15HSD17B10HPGDHDAC3
SCHEMBL9283660 0.78 TYR (0.47) ALDH1A1ALOX15HSD17B10HPGDMAPK1
SCHEMBL6273700 0.73 ESR1 (0.40) ALDH1A1ALOX15HSD17B10HPGDALOX12
SCHEMBL27909752 0.72 CYP3A4 (0.43) ALDH1A1ALOX15HSD17B10HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL9808420 0.71 ESR1 (0.39) ALDH1A1ALOX15HSD17B10HPGDALOX12
SCHEMBL7041926 0.71 KDM4E (0.40) ALDH1A1ALOX15HSD17B10MAPK1HDAC3
SCHEMBL9382243 0.71 IDO1 (0.47) ALDH1A1HSD17B10SMN1; SMN2MAPK1IDO1
SCHEMBL3838657 0.71 PRKCI (0.34) ALDH1A1GAAKDM4EPRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976861-A2 INHIBITING TUMOUR CELL INVASION, METASTASIS AND ANGIOGENESIS THROUGH TARGETTING LEGUMAIN The Scripps Research Institute (US) 2008-10-08 EP disclosed
WO-2007064759-A2 INHIBITING TUMOUR CELL INVASION, METASTASIS AND ANGIOGENESIS THROUGH TARGETTING LEGUMAIN THE SCRIPPS RESEARCH INSTITUTE (US) 2007-06-07 WO disclosed