SCHEMBL5133372

SCHEMBL5133372

Nc1ccc(N)c(CCCl)c1CCCl

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.32
TDP1 Q9NUW8 3/20 0.32
TSHR P16473 3/20 0.32
ALOX15 P16050 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
TP53 P04637 1/20 0.32
THRB P10828 1/20 0.32
SKP2 Q13309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7517167 0.97 CYP3A4 (0.33) CYP3A4TDP1TSHRALOX15SMN1; SMN2
SCHEMBL5082011 0.86 ALDH1A1 (0.35) CYP3A4TDP1ALOX15SMN1; SMN2ALDH1A1
SCHEMBL27909752 0.83 CYP3A4 (0.43) CYP3A4TDP1TSHRALOX15SMN1; SMN2
SCHEMBL9382243 0.82 IDO1 (0.47) CYP3A4TDP1TSHRSMN1; SMN2ALDH1A1
SCHEMBL3838657 0.82 PRKCI (0.34) ALDH1A1
SCHEMBL28216128 0.81 POLB (0.38) CYP3A4TDP1TSHRALOX15SMN1; SMN2
SCHEMBL28120010 0.81
SCHEMBL28297642 0.81 TDP1 (0.31) TDP1THRB
SCHEMBL27966908 0.81 KDM4E (0.34) CYP3A4TSHRALDH1A1
SCHEMBL3674257 0.79 NOS2 (0.33) SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106631874-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-acetyl group -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN claimed
CN-106631857-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-propiono -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN claimed
CN-106631874-A Arylamine nitrogen mustard derivative N,N-bis(2-chloroethyl)-N'-acetyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN claimed
CN-106631857-A Aryl nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-propionyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN claimed
CN-106631857-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-propiono -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN disclosed
CN-106631874-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-acetyl group -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN disclosed
CN-106631874-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-acetyl group -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN disclosed
CN-106631857-B Arylamine nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-propiono -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-10 CN disclosed
CN-106631876-B (2- the chloroethyl)-N '-myristoyl of nitrogen mustard derivatives N, N- bis- base-Isosorbide-5-Nitrae-phenylenediamine and preparation method thereof 长安大学 2019-05-03 CN disclosed
CN-106631876-B (2- the chloroethyl)-N '-myristoyl of nitrogen mustard derivatives N, N- bis- base-Isosorbide-5-Nitrae-phenylenediamine and preparation method thereof 长安大学 2019-05-03 CN disclosed
CN-106631875-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-hexadecanoyl group -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-03 CN disclosed
CN-106631875-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-hexadecanoyl group -1,4- phenylenediamine and preparation method thereof 长安大学 2019-05-03 CN disclosed
CN-106631856-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-benzoyl -1,4- phenylenediamine and preparation method thereof 长安大学 2019-03-19 CN disclosed
CN-106631856-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-benzoyl -1,4- phenylenediamine and preparation method thereof 长安大学 2019-03-19 CN disclosed
CN-106631876-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-myristoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631875-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-hexadecanoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631856-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-benzoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631857-A Aryl nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-propionyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631874-A Arylamine nitrogen mustard derivative N,N-bis(2-chloroethyl)-N'-acetyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
EP-1897561-A1 Polymeric prodrugs of amino- and hydroxyl-containing bioactive agents ENZON, INC. (US) 2008-03-12 EP disclosed