SCHEMBL5083235

SCHEMBL5083235

CCCCCN1CCC(c2ccccc2)C(COc2ccc(OC)cc2)C1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
DRD4 P21917 7/20 0.43
HTR1A P08908 6/20 0.43
DRD1 P21728 6/20 0.43
DRD5 P21918 6/20 0.43
DRD3 P35462 6/20 0.43
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
DRD2 P14416 7/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416521 0.91 KMT2A (0.45) KMT2ACHRM2CHRM4CHRM5CHRM1
SCHEMBL7416518 0.91 KMT2A (0.45) KMT2ACHRM2CHRM4CHRM5CHRM1
SCHEMBL7416523 0.91 KMT2A (0.45) KMT2ACHRM2CHRM4CHRM5CHRM1
SCHEMBL5076788 0.90 KDM4E (0.48) KMT2ADRD4HTR1ADRD1DRD5
SCHEMBL5083179 0.89 HTT (0.44) DRD4HTR1ADRD1DRD5DRD3
SCHEMBL5083196 0.89 HTT (0.44) DRD4HTR1ADRD1DRD5DRD3
SCHEMBL5083190 0.89 HTT (0.44) DRD4HTR1ADRD1DRD5DRD3
Hydrochloric Acid SCHEMBL1152994 0.89 HTT (0.43) DRD4HTR1ADRD1DRD5DRD3
SCHEMBL5141567 0.89 HTR1A (0.44) KMT2ADRD4HTR1ADRD1DRD5
Hydrochloric Acid SCHEMBL1152993 0.89 HTT (0.43) DRD4HTR1ADRD1DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008133884-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-11-06 WO disclosed
EP-0266574-B1 Piperidine compounds and their preparation and use NOVO NORDISK AS (DK) 1994-01-05 EP disclosed
US-5019582-A Preventing Calcium Overload In Brain Cells NOVO NORDISK A/S (DK) 1991-05-28 US disclosed
US-4985446-A CALCIUM OVERLOAD BLOCKERS IN BRAIN CELLS A/S FERROSAN (DK) 1991-01-15 US disclosed
US-4877799-A Method of treating calcium overload in brain cells of mammals A/S FERROSAN (DK) 1989-10-31 US disclosed