SCHEMBL5084818

SCHEMBL5084818

O=c1[nH]c(Cc2ccccc2)nc2nc[nH]c12

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PNP P00491 3/20 0.58
KMT2A Q03164 1/20 0.54
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
RNASEH1 O60930 1/20 0.49
DAO P14920 1/20 0.49
GRIA1 P42261 1/20 0.47
GRIA2 P42262 1/20 0.47
GRIA3 P42263 1/20 0.47
GRIA4 P48058 1/20 0.47
PDE5A O76074 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5677631 0.83 PNP (0.80) PNPKMT2ARNASEH1DAO
SCHEMBL3757599 0.82 PDE4A (0.49) PNPKMT2APDE4APDE4BPDE4C
SCHEMBL8509084 0.78 PNP (0.62) PNPGRIA1GRIA2GRIA3GRIA4
SCHEMBL28817761 0.77 ADORA3 (0.49) PNPKMT2APDE4APDE4BPDE4C
SCHEMBL3396585 0.76 PNP (0.57) PNPGRIA1GRIA2GRIA3GRIA4
SCHEMBL11133891 0.76 PNP (0.57) PNPGRIA1GRIA2GRIA3GRIA4
SCHEMBL3433603 0.76 TSHR (0.52) PNPKMT2AGRIA1GRIA2GRIA3
SCHEMBL3757591 0.76 CYP1A2 (0.68) DAO
SCHEMBL18251 0.76 PNP (0.62) PNPPDE4APDE4BPDE4CPDE4D
Guanine SCHEMBL1394087 0.75 PNP (0.68) PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104447746-A Compound for activating AMPK and application thereof HUAAN MEDICAL CO LTD 2015-03-25 CN claimed
WO-2008109417-A1 MGMT INHIBITOR COMBINATIONS FOR THE TREATMENT OF NEOPLASTIC DISORDERS CASE WESTERN RESERVE UNIVERSITY (US) 2008-09-12 WO claimed
CN-104447746-A Compound for activating AMPK and application thereof HUAAN MEDICAL CO LTD 2015-03-25 CN disclosed