SCHEMBL5094020

SCHEMBL5094020

Cc1cccc(C(=O)NCc2ccc(C(=N)N)cc2N)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
F10 P00742 3/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ATM Q13315 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
F2 P00734 2/20 0.45
F7 P08709 1/20 0.45
KLKB1 P03952 7/20 0.45
PRSS1 P07477 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5089093 0.99 CA1 (0.49) POLBCA1CA2F10NPC1
SCHEMBL5094014 0.89 CA1 (0.49) POLBCA1CA2F10NPC1
SCHEMBL5177698 0.84 ALDH1A1 (0.52) POLBCA1CA2F10PRSS1
Hydrochloric Acid SCHEMBL5086280 0.84 CA1 (0.43) POLBCA1CA2F10NPC1
SCHEMBL5564415 0.83 CA1 (0.44) POLBCA1CA2F10NPC1
SCHEMBL8266386 0.83 F10 (0.45) POLBCA1CA2F10NPC1
Hydrochloric Acid SCHEMBL5089718 0.83 ALDH1A1 (0.51) POLBCA1CA2PRSS1KDM4E
Hydrochloric Acid SCHEMBL5089572 0.82 CA1 (0.43) POLBCA1CA2F10NPC1
Hydrochloric Acid SCHEMBL5139096 0.82 F10 (0.46) POLBCA1CA2F10RAB9A
SCHEMBL8267082 0.82 HDAC8 (0.53) CA1CA2F10NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008512364-A 2008-04-24 JP claimed
EP-1791810-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIA INHIBITORS F. Hoffmann-Roche AG (CH) 2007-06-06 EP claimed
WO-2006027135-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIIA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-16 WO claimed
EP-1791810-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIA INHIBITORS F. Hoffmann-Roche AG (CH) 2007-06-06 EP disclosed
WO-2006027135-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIIA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-16 WO disclosed
WO-2006027135-A1 4-AMINOMETHYL BENZAMIDINE DERIVATIVES AND THEIR USE AS FACTOR VIIIA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-16 WO disclosed