SCHEMBL5120701

SCHEMBL5120701

FC(F)(F)c1cccc(-c2cncc(N3CCN4CC3C4)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.45
CYP11B1 P15538 1/20 0.45
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
MGLL Q99685 1/20 0.38
GRIN2B Q13224 7/20 0.38
GRIN1 Q05586 4/20 0.38
KDM1A O60341 1/20 0.37
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
NPY5R Q15761 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5116073 0.92 CYP11B1 (0.43) CYP11B2CYP11B1NR3C1PGRMGLL
Hydrochloric Acid SCHEMBL5123727 0.91 CYP11B1 (0.42) CYP11B2CYP11B1NR3C1PGRMGLL
SCHEMBL5110755 0.90 CYP11B1 (0.41) CYP11B2CYP11B1NR3C1PGRMGLL
SCHEMBL5108601 0.87 CYP11B1 (0.43) CYP11B2CYP11B1NR3C1PGRMGLL
SCHEMBL5115900 0.86 CHRNB4 (0.42) CYP11B2CYP11B1KDM1ACHRNB4CHRNA3
SCHEMBL5115363 0.85 CYP11B1 (0.41) CYP11B2CYP11B1NR3C1PGRMGLL
SCHEMBL5123104 0.82 CHRNB4 (0.52) CYP11B2CYP11B1CHRNB4CHRNA3
SCHEMBL5123133 0.81 CHRNB4 (0.39) CHRNB4CHRNA3HTR2AHTR2CHTR2B
SCHEMBL6836268 0.81 NR1H2 (0.43) CYP11B2CYP11B1CHRNB4CHRNA3HTR2A
SCHEMBL5115818 0.79 HDAC8 (0.44) NR3C1PGRMGLLGRIN2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040106603-A1 Diazabicyclic compounds useful in the treatment of CNS and other disorders PFIZER INC 2004-06-03 US claimed
US-7442694-B2 Diazabicyclic compounds useful in the treatment of CNS and other disorders PFIZER INC (US) 2008-10-28 US disclosed
US-20040106603-A1 Diazabicyclic compounds useful in the treatment of CNS and other disorders PFIZER INC 2004-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040106603-A1 Diazabicyclic compounds useful in the treatment of CNS and other disorders DBH, CHRNA6, DDT CYP11B2 403/4885CYP11B1 273/4885NR3C1 149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.