SCHEMBL5127768

SCHEMBL5127768

Fc1ccc(-c2ccc3ncnc(OC4CCCC4)c3c2)cc1.Fc1ccc(-c2ccc3ncnc(OCc4ccccc4)c3c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK1 P51617 1/20 0.49
IRAK4 Q9NWZ3 1/20 0.49
LMNA P02545 3/20 0.42
PIK3CD O00329 6/20 0.42
PIK3CA P42336 5/20 0.42
PIK3CB P42338 5/20 0.42
PIK3CG P48736 5/20 0.42
MAP4K4 O95819 2/20 0.42
CAMKK1 Q8N5S9 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
DHODH Q02127 1/20 0.39
KCNH2 Q12809 2/20 0.39
SCN5A Q14524 2/20 0.39
SCN9A Q15858 2/20 0.39
KDR P35968 1/20 0.39
RAF1 P04049 1/20 0.38
BRAF P15056 1/20 0.38
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3334180 0.88 MAP4K4 (0.52) LMNAMAP4K4DHODHKDRRAF1
SCHEMBL3336126 0.88 MAP4K4 (0.52) IRAK4PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL5131672 0.83 RAB9A (0.49) IRAK1IRAK4PIK3CDPIK3CAPIK3CB
SCHEMBL3336037 0.74 MAP4K4 (0.52) IRAK4LMNAPIK3CDPIK3CAPIK3CB
SCHEMBL3335725 0.72 MAP4K4 (0.41) PIK3CAMAP4K4SCN9A
SCHEMBL3334604 0.72 ADORA2A (0.50) LMNAMAP4K4DHODHSCN9ACYP1A2
SCHEMBL3336424 0.71 PIK3CD (0.53) IRAK1IRAK4LMNAPIK3CDPIK3CA
SCHEMBL3332824 0.71 PIK3CD (0.74) IRAK1IRAK4PIK3CDPIK3CAPIK3CB
SCHEMBL3334866 0.71 MAP4K4 (0.57) LMNAMAP4K4RAF1BRAFUSP2
SCHEMBL3333219 0.69 PIK3CD (0.51) IRAK4LMNAPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed