SCHEMBL5131672

SCHEMBL5131672

CC(=O)Nc1ccc(-c2ccc3ncnc(OC4CCCC4)c3c2)cc1.CC(=O)Nc1ccc(-c2ccc3ncnc(OCc4ccccc4)c3c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.49
IRAK1 P51617 1/20 0.46
IRAK4 Q9NWZ3 1/20 0.46
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
PIK3CD O00329 4/20 0.43
PIK3CA P42336 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
JAK2 O60674 1/20 0.43
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
MAP4K4 O95819 1/20 0.43
C5AR1 P21730 1/20 0.42
FDPS P14324 1/20 0.42
ACACB O00763 1/20 0.42
PPIA P62937 1/20 0.41
TSHR P16473 1/20 0.41
MAP3K8 P41279 1/20 0.41
CAMKK1 Q8N5S9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3333219 0.90 PIK3CD (0.51) RAB9AIRAK4PIK3CDPIK3CAPIK3CB
SCHEMBL3335286 0.90 RAB9A (0.56) RAB9ACYP11B1CYP11B2JAK2RAF1
SCHEMBL5127768 0.83 IRAK1 (0.49) IRAK1IRAK4PIK3CDPIK3CAPIK3CB
SCHEMBL3337576 0.78 RAB9A (0.51) RAB9APIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3334949 0.77 BRAF (0.43) RAB9ABRAFKDM4EMEN1KMT2A
SCHEMBL3340079 0.77 JAK2 (0.47) CYP11B1CYP11B2PIK3CAJAK2BRAF
SCHEMBL5127968 0.77 CNR1 (0.35) CYP11B1CYP11B2JAK2ACACBPPIA
SCHEMBL3338478 0.77 RAB9A (0.56) RAB9ARAF1BRAFMAP4K4MAP3K8
SCHEMBL3341282 0.77 GHSR (0.54) CYP11B1CYP11B2JAK2MAP4K4FDPS
SCHEMBL3337132 0.77 CYP2D6 (0.42) RAB9AMAP4K4KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed