SCHEMBL5129448

SCHEMBL5129448

CC(=O)Nc1ccc(-c2ccc3nc(NC(C)=O)nc(OCc4ccccc4)c3c2)cc1.CCCOc1nc(NC(C)=O)nc2ccc(-c3ccc(NC(C)=O)cc3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.43
FDPS P14324 1/20 0.42
MOK Q9UQ07 3/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
TSHR P16473 1/20 0.42
PPIA P62937 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
GHSR Q92847 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
KDM4E B2RXH2 3/20 0.41
BRAF P15056 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TP53 P04637 1/20 0.41
APP P05067 1/20 0.41
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340079 0.94 JAK2 (0.47) JAK2FDPSCYP11B1CYP11B2TSHR
SCHEMBL3339894 0.92 BRAF (0.47) FDPSMOKMEN1KMT2AKDM4E
SCHEMBL5129183 0.90 GHSR (0.49) JAK2FDPSMOKCYP11B1CYP11B2
SCHEMBL3336607 0.87 BRAF (0.46) FDPSMOKTDP1MEN1KMT2A
SCHEMBL3334534 0.85 DHODH (0.48) KDM4EALDH1A1HPGDAPPACHE
SCHEMBL3331750 0.84 TTK (0.48) FDPSMOKTDP1MEN1KMT2A
SCHEMBL3341282 0.83 GHSR (0.54) JAK2FDPSCYP11B1CYP11B2TSHR
SCHEMBL3335706 0.83 NAMPT (0.42) KDM4EBRAFALDH1A1MAPTHPGD
SCHEMBL3336288 0.83 MOK (0.47) FDPSMOKMEN1KMT2AKDM4E
SCHEMBL3338586 0.82 ACHE (0.54) TSHRTDP1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed