SCHEMBL5131652

SCHEMBL5131652

CCOc1nc(N)nc2ccc(-c3ccc(C(=O)N4CCCCC4)cc3)cc12.CNC(=O)c1cccc(-c2ccc3nc(N)nc(OCC4CC4)c3c2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRIM58 Q8NG06 1/20 0.41
DCPS Q96C86 1/20 0.40
CHEK2 O96017 1/20 0.40
MGLL Q99685 1/20 0.40
BRD4 O60885 1/20 0.39
CNR2 P34972 2/20 0.39
POLB P06746 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SCN9A Q15858 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
PDE4D Q08499 1/20 0.38
HPGD P15428 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5129519 0.89 MGLL (0.40) MGLLPOLBHPGDADORA2AADORA1
SCHEMBL3340183 0.87 TRIM58 (0.50) TRIM58CNR2SCN9AAKT1AKT2
SCHEMBL3336761 0.84 HPGD (0.51) MGLLL3MBTL1HPGD
SCHEMBL3335650 0.83 HPGD (0.50) MGLLL3MBTL1HPGD
SCHEMBL3335317 0.82 MAP4K4 (0.48)
SCHEMBL3336243 0.81 TRIM58 (0.48) TRIM58AKT1AKT2
SCHEMBL3338030 0.78 PLK1 (0.46)
SCHEMBL5127579 0.78 HPGD (0.44) MGLLL3MBTL1HPGD
SCHEMBL3336878 0.76 TRIM58 (0.46) TRIM58CNR2PDE4D
SCHEMBL3333969 0.76 HPGD (0.43) MGLLPOLBL3MBTL1HPGDADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed