SCHEMBL5131696

SCHEMBL5131696

CC(=O)Nc1ccc(-c2ccc3nc(NC(C)=O)nc(OC(F)(F)F)c3c2)cc1.CC(=O)Nc1ccc(-c2ccc3nc(NC(C)=O)nc(OCC(F)(F)F)c3c2)cc1.CC(=O)Nc1ccc(-c2ccc3nc(NC(C)=O)nc(OCC4CC4)c3c2)cc1.CCOc1nc(NC(C)=O)nc2ccc(-c3ccc(NC(C)=O)cc3)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM58 Q8NG06 1/20 0.47
HTR2A P28223 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTR4 Q13639 1/20 0.39
SYK P43405 2/20 0.37
NPR1 P16066 1/20 0.35
TTK P33981 1/20 0.35
MAPK8 P45983 1/20 0.35
BRAF P15056 1/20 0.35
CDK12 Q9NYV4 1/20 0.35
CNR2 P34972 2/20 0.34
PIK3CA P42336 1/20 0.34
CNR1 P21554 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
CTPS1 P17812 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34
PAX8 Q06710 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3337025 0.86 TRIM58 (0.56) TRIM58HTR2AKCNH2HTR4NPR1
SCHEMBL5179372 0.85 TRIM58 (0.41) TRIM58HTR2AKCNH2HTR4SYK
SCHEMBL3335653 0.85 SYK (0.45) TRIM58SYKTTKMAPK8BRAF
SCHEMBL3333273 0.82 KMT2A (0.47) SYKBRAFPIK3CAMEN1LMNA
SCHEMBL3331750 0.81 TTK (0.48) TTKMAPK8BRAFMEN1LMNA
SCHEMBL3333859 0.80 TRIM58 (0.55) TRIM58HTR2AKCNH2HTR4NPR1
SCHEMBL3341530 0.78 PIK3CA (0.44) TRIM58SYKBRAFPIK3CAMEN1
SCHEMBL3337337 0.76 TRIM58 (0.48) TRIM58HTR2AKCNH2HTR4BRAF
SCHEMBL5131263 0.76 KCNH2 (0.44) TRIM58HTR2AKCNH2HTR4CNR2
SCHEMBL3340067 0.75 MAPK10 (0.43) SYKBRAFPIK3CAMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009077-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed