SCHEMBL5132284

SCHEMBL5132284

O=C(O)c1cn2c(c(O)c1=O)C(=O)N(CCOc1ccccc1)CC2

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.40
KCNA5 P22460 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20015178 0.84 ITGB3 (0.38)
SCHEMBL2184756 0.82 PTPN7 (0.45) KMT2A
SCHEMBL20014841 0.82 ITGB3 (0.35)
SCHEMBL20014376 0.80 LMNA (0.46) NPC1RAB9AKMT2APOLB
SCHEMBL20014654 0.80 HTT (0.46)
SCHEMBL20014699 0.79 ITGB3 (0.35)
SCHEMBL20014364 0.77 KDM4E (0.37) MEN1KMT2AALDH1A1
SCHEMBL23341013 0.77 ITGB3 (0.36)
SCHEMBL20015188 0.74 ITGB3 (0.37)
SCHEMBL5132211 0.73 AKR1B1 (0.45) RAB9AMEN1KMT2APOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1950212-B1 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING INHIBITORY ACTIVITY ON HIV INTEGRASE SHIONOGI & CO (JP) 2016-02-24 EP disclosed
EP-1950212-A1 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING INHIBITORY ACTIVITY ON HIV INTEGRASE Shionogi Co., Ltd. (JP) 2008-07-30 EP disclosed