SCHEMBL5133166

SCHEMBL5133166

CC(C(=O)NO)C1=CCN(CCc2ccccc2F)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SLC1A2 P43004 1/20 0.41
DAO P14920 1/20 0.37
XIAP P98170 1/20 0.36
BIRC2 Q13490 1/20 0.36
HTR2A P28223 2/20 0.36
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2568713 0.75 HDAC3 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2565221 0.72 HDAC3 (0.42) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL5133163 0.70 OPRM1 (0.41) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL27650886 0.69 HDAC3 (0.41) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL6077832 0.63 LIPG (0.44) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL6297593 0.60 TAAR1 (0.48) ALDH1A1MEN1KMT2ASLC1A2TAAR1
SCHEMBL5871311 0.60 TACR1 (0.48) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL2905073 0.59 SLC1A2 (0.65) ALDH1A1SLC1A2TSHRLMNAHPGD
Hydrochloric Acid SCHEMBL22607752 0.59 SIRT2 (0.46) ALDH1A1CYP1A2CYP2C19KMT2AHTR2A
SCHEMBL27728237 0.58 TSHR (0.46) ALDH1A1MEN1KMT2ATAAR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1626961-A4 NOVEL 2-OXO-HETEROCYCLIC COMPOUNDS AND THE PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME KOREA RES INST OF BIOSCIENCE (KR) 2008-07-16 EP disclosed
EP-1626961-A1 NOVEL 2-OXO-HETEROCYCLIC COMPOUNDS AND THE PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Korea Research Institute of Bioscience and Biotechnology (KR) 2006-02-22 EP disclosed
WO-2004101523-A1 NOVEL 2-OXO-HETEROCYCLIC COMPOUNDS AND THE PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY (KR) 2004-11-25 WO disclosed