SCHEMBL5134048

SCHEMBL5134048

COc1ccc2c(c1)N(CCN1CC[CH]CC1)C(=O)OC2

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.55
KDM1A O60341 1/20 0.42
UBE2I P63279 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
OXTR P30559 3/20 0.38
HTR2A P28223 1/20 0.37
CHRM1 P11229 1/20 0.36
NQO2 P16083 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708467 0.85 KCNH2 (0.57) KCNH2KDM1AUBE2IHKDC1SAE1
SCHEMBL921899 0.80 KCNH2 (0.59) KCNH2UBE2IHKDC1SAE1UBA2
SCHEMBL705556 0.80 KCNH2 (0.52) KCNH2UBE2IHKDC1SAE1UBA2
Trifluoroacetic Acid SCHEMBL705051 0.78 KCNH2 (0.51) KCNH2UBE2IHKDC1SAE1UBA2
Trifluoroacetic Acid SCHEMBL704661 0.74 KCNH2 (0.43) KCNH2CHRM1
SCHEMBL706058 0.73 KCNH2 (1.00) KCNH2
SCHEMBL706037 0.70 KCNH2 (0.70) KCNH2HTR2A
SCHEMBL6602559 0.67 LMNA (0.49) OXTRKDM4EHSD17B10
SCHEMBL30293275 0.67 LMNA (0.49) OXTRKDM4EHSD17B10
SCHEMBL31033195 0.67 ALDH1A1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893599-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS AstraZeneca AB (SE) 2008-03-05 EP disclosed
WO-2006134378-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2006-12-21 WO disclosed