SCHEMBL5134328

SCHEMBL5134328

CN(C(=O)c1ccc(Oc2ccccc2)cc1CC1CCCO1)C1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.48
SLC6A4 P31645 6/20 0.48
KCNH2 Q12809 5/20 0.48
RAB9A P51151 2/20 0.46
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
OXTR P30559 2/20 0.40
AVPR1A P37288 2/20 0.40
HPGD P15428 4/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SLC6A3 Q01959 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135114 0.81 SLC6A2 (0.53) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL8738173 0.73 SLC6A4 (0.59) SLC6A2SLC6A4KCNH2RAB9AMEN1
SCHEMBL5146827 0.71 CNR2 (0.41) SLC6A2SLC6A4HPGDSLC6A3CYP2D6
SCHEMBL5134331 0.70 RAB9A (0.39) SLC6A2SLC6A4RAB9AMEN1KMT2A
SCHEMBL5134122 0.69 PARP1 (0.41) KCNH2KMT2ALMNASMN1; SMN2OXTR
Trifluoroacetic Acid SCHEMBL6119832 0.68 SLC6A4 (0.53) SLC6A2SLC6A4KCNH2MEN1KMT2A
SCHEMBL28093969 0.67 ALOX5 (0.45) RAB9A
SCHEMBL5136170 0.66 SLC6A4 (0.44) SLC6A2SLC6A4KCNH2RAB9AHPGD
SCHEMBL4109434 0.65 SLC6A4 (1.00) SLC6A2SLC6A4KCNH2LMNASLC6A3
SCHEMBL4651364 0.65 CACNA1B (0.47) SLC6A2SLC6A4KCNH2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed