SCHEMBL5134527

SCHEMBL5134527

CN(C(=O)c1ccc(F)c(CC2CCOCC2)c1F)C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.39
PARP1 P09874 1/20 0.39
SLC6A2 P23975 7/20 0.38
KCNH2 Q12809 5/20 0.38
SLC6A3 Q01959 4/20 0.38
CYP2D6 P10635 2/20 0.38
HSD11B1 P28845 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
KIF11 P52732 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135452 0.82 SLC6A4 (0.47) SLC6A4PARP1SLC6A2KCNH2SLC6A3
SCHEMBL5140427 0.81 SLC6A4 (0.38) SLC6A4SLC6A2KCNH2SLC6A3CYP2D6
SCHEMBL5190868 0.75 SLC6A4 (0.45) SLC6A4SLC6A2KCNH2SLC6A3CYP2D6
SCHEMBL5146827 0.73 CNR2 (0.41) SLC6A4PARP1SLC6A2SLC6A3CYP2D6
SCHEMBL5136170 0.72 SLC6A4 (0.44) SLC6A4SLC6A2KCNH2SLC6A3CYP2D6
SCHEMBL5134802 0.71 PARP1 (0.51) SLC6A4PARP1SLC6A2KCNH2SLC6A3
SCHEMBL5134122 0.70 PARP1 (0.41) PARP1KCNH2KMT2AKDM4EPOLB
SCHEMBL19710924 0.67 PDK2 (0.50) HSD11B1KMT2AMEN1RAB9AKDM4E
SCHEMBL28633494 0.66 SMO (0.53) SLC6A4SLC6A2SLC6A3KMT2A
SCHEMBL5134854 0.65 CNR1 (0.37) PARP1KCNH2KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed