SCHEMBL5134802

SCHEMBL5134802

CN(C(=O)c1cc(F)ccc1F)C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.51
KCNH2 Q12809 4/20 0.47
KIF11 P52732 2/20 0.47
SLC6A4 P31645 8/20 0.46
SLC6A2 P23975 6/20 0.46
CES2 O00748 2/20 0.45
CES1 P23141 2/20 0.45
SLC6A3 Q01959 3/20 0.45
DPP4 P27487 3/20 0.42
DPP9 Q86TI2 3/20 0.42
DPP7 Q9UHL4 3/20 0.42
DPP8 Q6V1X1 2/20 0.42
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633494 0.82 SMO (0.53) SLC6A4SLC6A2SLC6A3
SCHEMBL28646233 0.81 CCR5 (0.51) KCNH2KIF11SLC6A4SLC6A2SLC6A3
SCHEMBL30323082 0.77 CES2 (0.52) CES2CES1
SCHEMBL20524724 0.77 CES2 (0.52) CES2CES1
Hydrochloric Acid SCHEMBL15567881 0.76 CES2 (0.50) CES2CES1
Hydrochloric Acid SCHEMBL31196625 0.76 CES2 (0.50) CES2CES1
SCHEMBL31270828 0.74 CES2 (0.61) CES2CES1TAS1R3TAS1R1TAS1R2
SCHEMBL8566777 0.74 CES2 (0.61) CES2CES1TAS1R3TAS1R1TAS1R2
SCHEMBL10107580 0.73 SLC6A4 (0.64) KCNH2SLC6A4SLC6A2SLC6A3
SCHEMBL4154297 0.72 HPGD (0.54) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1901746-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2008-03-26 EP disclosed
WO-2007002884-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-01-04 WO disclosed