SCHEMBL5190868

SCHEMBL5190868

Cc1c(CC2CCOCC2)cccc1C(=O)N(C)C1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.45
SLC6A2 P23975 13/20 0.43
SLC6A3 Q01959 9/20 0.43
CYP2D6 P10635 6/20 0.43
HSD11B1 P28845 1/20 0.42
KCNH2 Q12809 4/20 0.40
CHRM1 P11229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136170 0.83 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3CYP2D6HSD11B1
SCHEMBL5135452 0.83 SLC6A4 (0.47) SLC6A4SLC6A2SLC6A3CYP2D6HSD11B1
SCHEMBL5134527 0.75 SLC6A4 (0.39) SLC6A4SLC6A2SLC6A3CYP2D6HSD11B1
SCHEMBL5140427 0.74 SLC6A4 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6HSD11B1
SCHEMBL16099881 0.69 HSD11B1 (0.53) SLC6A4SLC6A2SLC6A3HSD11B1KCNH2
SCHEMBL23228615 0.67 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3
SCHEMBL10107580 0.66 SLC6A4 (0.64) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL12209651 0.66 HTR2C (0.45) HSD11B1
SCHEMBL3969439 0.66 HTR2C (0.53) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL4291607 0.65 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed