SCHEMBL5134598

SCHEMBL5134598

CCCc1nn(C)c2cnc(NCc3ccc4c(ccn4C)c3)nc12

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.39
PDE5A O76074 1/20 0.38
CLK4 Q9HAZ1 4/20 0.37
CACNA1H O95180 4/20 0.35
CHRNA7 P36544 7/20 0.35
PIK3CB P42338 1/20 0.34
PTK2 Q05397 1/20 0.34
PTK2B Q14289 1/20 0.34
AURKA O14965 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134154 0.76 CCNA2 (0.48) PTK2AURKA
SCHEMBL4900033 0.75 PDE5A (0.48) PDE5A
SCHEMBL5134597 0.75 PIK3CB (0.34) PIK3CB
SCHEMBL5133695 0.72 PDE10A (0.41) PDE5ACLK4
SCHEMBL18876154 0.69 PRKCI (0.52) TRPV1CACNA1HCHRNA7PIK3CB
SCHEMBL5134599 0.68 MKNK1 (0.40)
SCHEMBL4897814 0.67 PDE5A (0.48) PDE5A
SCHEMBL3122462 0.66 PDE5A (0.36) PDE5A
SCHEMBL1253366 0.66 CHRNA7 (0.50) TRPV1CHRNA7
SCHEMBL10111229 0.64 PRKCI (0.49) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO claimed
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO disclosed