SCHEMBL5134607

SCHEMBL5134607

CCCc1nn(C)c2cnc(N(C)Cc3ccc(-c4cncnc4)cc3)nc12

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.33
HDAC1 Q13547 1/20 0.32
RPS6KB1 P23443 2/20 0.31
JAK1 P23458 1/20 0.31
NMT1 P30419 1/20 0.31
PDE5A O76074 2/20 0.31
HDAC6 Q9UBN7 1/20 0.30
ICMT O60725 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133891 0.81 NMT1 (0.42) HDAC1NMT1PDE5AHDAC6
SCHEMBL4901866 0.75 PDE5A (0.51) ALDH1A1HDAC1PDE5AHDAC6
SCHEMBL5134315 0.68 PDE5A (0.35) LMNASMN1; SMN2ALDH1A1PDE5A
SCHEMBL4137516 0.66 LMNA (0.31) LMNA
SCHEMBL4893654 0.66 PDE5A (0.52) ALDH1A1HDAC1PDE5AHDAC6
SCHEMBL3122462 0.66 PDE5A (0.36) LMNASMN1; SMN2ALDH1A1PDE5A
SCHEMBL4904011 0.65 PDE5A (0.52) ALDH1A1HDAC1NMT1PDE5AHDAC6
SCHEMBL13988124 0.64 ATM (0.46) SMN1; SMN2HDAC1
SCHEMBL5134598 0.62 TRPV1 (0.39) PDE5A
SCHEMBL4903930 0.60 PDE5A (0.52) ALDH1A1HDAC1PDE5AHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO claimed
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO disclosed