SCHEMBL5134689

SCHEMBL5134689

CCCc1nn(C)c2cnc(N(Cc3cccc(N4CCOCC4)c3)CC(C)C)nc12

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.35
AGXT P21549 1/20 0.34
HDAC1 Q13547 1/20 0.33
PIK3R2 O00459 5/20 0.33
ALKBH1 Q13686 1/20 0.32
BRD4 O60885 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TRPV3 Q8NET8 1/20 0.32
LCK P06239 1/20 0.32
KDR P35968 1/20 0.32
DHFR P00374 1/20 0.32
HTR1A P08908 1/20 0.32
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
KDM5B Q9UGL1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134147 0.80 RORC (0.34) RORCAGXTALKBH1LCKKDR
SCHEMBL4901484 0.79 PDE5A (0.42) HDAC1HTR1A
SCHEMBL5134311 0.74 GBA1 (0.32)
SCHEMBL4905752 0.73 PDE5A (0.41) HDAC1HTR1A
SCHEMBL4901853 0.72 PDE5A (0.40) HDAC1HTR1A
SCHEMBL4895854 0.71 PDE5A (0.45) HDAC1HTR1A
SCHEMBL4142910 0.70 HSP90AA1 (0.37) AGXTHTR1AHTR1DHTR1B
SCHEMBL4892978 0.69 PDE5A (0.45) HDAC1HTR1A
SCHEMBL4901618 0.68 PDE5A (0.41) HDAC1HTR1A
SCHEMBL4128912 0.68 PDE5A (0.41) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO claimed
WO-2008071650-A2 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-06-19 WO disclosed