SCHEMBL4142910

SCHEMBL4142910

CCCc1n[nH]c2cnc(N(Cc3cccc(N4CCOCC4)c3)CC3CCCCC3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.37
HSP90AB1 P08238 5/20 0.37
TTK P33981 3/20 0.34
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
CTSL P07711 2/20 0.33
AGXT P21549 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
NAPEPLD Q6IQ20 1/20 0.32
FGFR1 P11362 1/20 0.32
FGFR2 P21802 1/20 0.32
FGFR3 P22607 1/20 0.32
ACVR1 Q04771 1/20 0.32
PRKDC P78527 1/20 0.32
CDC7 O00311 1/20 0.32
PLK4 O00444 1/20 0.32
MAP4K1 Q92918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8032543 0.81 HSP90AA1 (0.35) HSP90AA1HSP90AB1TTKAGXTPRKDC
SCHEMBL4123059 0.74 PDE5A (0.34) TTKPRKDC
SCHEMBL4287197 0.73 AGXT (0.37) TTKHTR1AHTR1DHTR1BCTSL
SCHEMBL4128912 0.73 PDE5A (0.41)
SCHEMBL5134689 0.70 RORC (0.35) HTR1AHTR1DHTR1BAGXT
SCHEMBL4282621 0.68 AGXT (0.36) TTKHTR1AHTR1DHTR1BCTSL
SCHEMBL4285889 0.67 AGXT (0.38) HTR1AHTR1DHTR1BCTSLAGXT
SCHEMBL4133677 0.66 TPH1 (0.33) AGXTPRKDC
SCHEMBL4128842 0.66 KDM4E (0.35) HTR1AHTR1DHTR1BAGXTPRKDC
SCHEMBL8032549 0.65 PDE5A (0.36) HTR1AHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071706-A1 PYRAZOLEPYRIMIDINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed