SCHEMBL5135645

SCHEMBL5135645

CCCCn1c(CN(Cc2ccc(OC)cc2)Cc2ccc(C(=O)O)cc2)cnc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 7/20 0.44
PTGES O14684 1/20 0.43
TAS2R8 Q9NYW2 1/20 0.43
CXCR3 P49682 1/20 0.43
LPAR1 Q92633 4/20 0.41
LPAR5 Q9H1C0 4/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PTPN1 P18031 1/20 0.41
ACHE P22303 1/20 0.40
PLA2G4A P47712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135023 0.93 AGTR1 (0.45) LPAR1LPAR5IRAK4SMN1; SMN2ACHE
SCHEMBL5138093 0.91 TSHR (0.43) NPC1RAB9ASMN1; SMN2
SCHEMBL5072318 0.90 TSHR (0.40) RAB9ASMN1; SMN2PTPN1
SCHEMBL5134636 0.87 AGTR1 (0.46)
SCHEMBL5134787 0.85 BCHE (0.42)
SCHEMBL5136085 0.84 AGTR1 (0.45) LPAR1LPAR5RAB9ASMN1; SMN2
SCHEMBL5135900 0.84 TLR7 (0.42) NPC1RAB9ASMN1; SMN2
SCHEMBL14415595 0.83 HPGD (0.44) RAB9ASMN1; SMN2
SCHEMBL5135175 0.83 AGTR1 (0.43) LPAR1LPAR5RAB9ASMN1; SMN2
SCHEMBL5134565 0.83 PPARG (0.42) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed