SCHEMBL5137573

SCHEMBL5137573

CCCCC(c1cnc(-c2ccccc2)n1CCCC)N(CCCC)Cc1ccc(OC)c(C(=O)OC)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 14/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136872 0.94 LMNA (0.40) CXCR3LMNAMEN1POLBKMT2A
SCHEMBL5135244 0.91 KDM4E (0.35) CXCR3LMNAMEN1POLBKMT2A
SCHEMBL650145 0.87 LPAR1 (0.40) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL5135309 0.86 TLR7 (0.41)
SCHEMBL5135388 0.86 CXCR3 (0.38) CXCR3LMNAMEN1POLBKMT2A
SCHEMBL5136929 0.86 LTB4R2 (0.37) LMNAMEN1POLBKMT2ATDP1
SCHEMBL5071417 0.82 TSHR (0.39) LMNAALDH1A1SMN1; SMN2
SCHEMBL5137622 0.82 CXCR3 (0.44) CXCR3
SCHEMBL5135939 0.82 HSP90AA1 (0.38)
SCHEMBL5136262 0.81 TLR7 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed