SCHEMBL5137967

SCHEMBL5137967

CN1C=CC=C(C(=O)Nc2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.41
HSD17B10 Q99714 2/20 0.41
NAPRT Q6XQN6 1/20 0.41
PKM P14618 1/20 0.40
ALDH1A1 P00352 5/20 0.40
POLB P06746 3/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 2/20 0.40
PTPN1 P18031 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12247923 0.76 HPGD (0.51) HPGDHSD17B10NAPRTALDH1A1POLB
SCHEMBL468058 0.75 TSHR (0.37) HSD17B10KMT2A
SCHEMBL28702490 0.75 TSHR (0.37) HSD17B10KMT2A
Water SCHEMBL28685341 0.73 TSHR (0.36) HSD17B10KMT2A
Iodide SCHEMBL21082066 0.72 CHRNB2 (0.40) ALDH1A1POLBKMT2AMEN1NPC1
SCHEMBL18250666 0.70 PTPN1 (0.43) HPGDHSD17B10NAPRTALDH1A1POLB
Iodide SCHEMBL9763182 0.70 NAMPT (0.36) ALDH1A1KMT2AMEN1NPC1RAB9A
Iodide SCHEMBL28802571 0.69 CHRM3 (0.45) POLBKDM4EPTPN1LMNAGAA
Iodide SCHEMBL3065810 0.68 GABRR1 (0.33) HSD17B10KMT2A
SCHEMBL12562736 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919466-A2 FORMULATIONS FOR TREATMENT OF LIPOPROTEIN ABNORMALITIES COMPRISING A STATIN AND A METHYLNICOTINAMIDE DERIVATIVE PHARMENA NORTH AMERICA INC. (CA) 2008-05-14 EP disclosed
WO-2007074406-A2 FORMULATIONS FOR TREATMENT OF LIPOPROTEIN ABNORMALITIES COMPRISING A STATIN A STATIN AND A METHYLNICOTINAMIDE DERIVATIVE PHARMENA NORTH AMERICA INC. (CA) 2007-07-05 WO disclosed