SCHEMBL5138866

SCHEMBL5138866

COc1cc(C(OC)n2ccc3cccnc32)ccc1OCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
CSF1R P07333 2/20 0.42
KMT2A Q03164 2/20 0.41
HPGD P15428 3/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5322845 0.77 CSF1R (0.55) LMNACSF1RKMT2AALDH1A1TSHR
SCHEMBL12738664 0.71 NPC1 (0.55) KMT2AHPGDALDH1A1TSHRHTT
SCHEMBL19734616 0.70 NPC1 (0.57) KMT2AHPGDALDH1A1HTTKDM4E
SCHEMBL14168120 0.70 NPC1 (0.57) KMT2AHPGDALDH1A1HTTKDM4E
SCHEMBL14167832 0.70 MEN1 (0.54) KMT2AHPGDALDH1A1TSHRHTT
SCHEMBL7369453 0.69 CTSV (0.50) KMT2AHPGDMEN1POLBGAA
SCHEMBL30806026 0.69 NPC1 (0.52) KMT2AHPGDALDH1A1HTTKDM4E
SCHEMBL28344001 0.69 NPC1 (0.56) KMT2AHPGDALDH1A1HTTKDM4E
SCHEMBL6375554 0.69 NPC1 (0.52) KMT2AHPGDALDH1A1HTTKDM4E
SCHEMBL28344002 0.69 NPC1 (0.56) KMT2AHPGDALDH1A1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893612-A1 PYRROLO [2, 3-B]PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2008-03-05 EP disclosed
WO-2007002433-A1 PYRROLO [2, 3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-01-04 WO disclosed