SCHEMBL5138874

SCHEMBL5138874

NC(=O)N(CCCCN1CCN(c2ccc3c(c2)OCCO3)CC1)c1cc2cc(Br)ccc2o1.NC(=O)Nc1cc2ccccc2n1CCCCN1CCN(c2ccc3c(c2)OCCO3)CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.41
DRD3 P35462 6/20 0.39
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
HTR1A P08908 4/20 0.35
OPRK1 P41145 1/20 0.35
HTR2A P28223 3/20 0.35
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
POLB P06746 1/20 0.34
HTR2C P28335 2/20 0.34
KCNH2 Q12809 2/20 0.34
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4952355 0.88 DRD2 (0.43) SLC6A4DRD3DRD2DRD4HTR1A
SCHEMBL5088731 0.87 DRD2 (0.41) DRD3DRD2DRD4HTR1AHTR2A
SCHEMBL4947889 0.85 DRD2 (0.41) SLC6A4DRD3DRD2DRD4HTR1A
SCHEMBL4950127 0.85 DRD2 (0.42) SLC6A4DRD3DRD2DRD4HTR1A
SCHEMBL4948673 0.84 SLC6A4 (0.53) SLC6A4DRD3DRD2HTR1AOPRK1
SCHEMBL4950273 0.84 ADRA2A (0.45) SLC6A4DRD3DRD2DRD4HTR1A
SCHEMBL4947477 0.82 DRD3 (0.47) SLC6A4DRD3DRD2HTR1AHTR2A
SCHEMBL4949597 0.82 SLC6A4 (0.50) SLC6A4DRD3DRD2HTR1AOPRK1
SCHEMBL4949782 0.81 SLC6A4 (0.49) SLC6A4DRD3DRD2HTR1AOPRK1
SCHEMBL4952129 0.80 SLC6A2 (0.41) SLC6A4DRD3DRD2DRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008526700-A 2008-07-24 JP claimed
EP-1761524-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2007-03-14 EP claimed
WO-2006072430-A1 PHENYL DIAZEPANE CARBOXAMIDES AND ANNELATED PHENYL PIPERAZINE CARBOXAMIDES CONTAINING OXYGEN AND USED AS DOPAMINE D3 ANTAGONISTS SCHWARZ PHARMA AG (DE) 2006-07-13 WO claimed