SCHEMBL5138974

SCHEMBL5138974

N#Cc1c(N)nc2cnccc2c1-c1ccccc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.53
ALDH1A1 P00352 6/20 0.53
GAA P10253 3/20 0.53
HPGD P15428 3/20 0.53
GLA P06280 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HSD17B10 Q99714 3/20 0.49
MAPK1 P28482 2/20 0.49
F7 P08709 2/20 0.46
F3 P13726 2/20 0.46
F10 P00742 1/20 0.46
PIP4K2A P48426 2/20 0.45
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
PDE10A Q9Y233 1/20 0.42
HTT P42858 1/20 0.41
IKBKB O14920 1/20 0.40
DHODH Q02127 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072774 0.85 ALDH1A1 (0.54) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL5138971 0.80 PIP4K2A (0.58) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6222236 0.78 SMN1; SMN2 (0.50) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6223236 0.77 ADORA1 (0.50) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6250192 0.71 KDM4E (0.69) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL7018457 0.71 ALDH1A1 (0.64) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL7024723 0.71 ALDH1A1 (0.67) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL6072338 0.70 KDM4E (0.62) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL28746020 0.70 RXFP1 (0.67) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL7018672 0.70 ALDH1A1 (0.72) KDM4EALDH1A1GAAHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7432279-B2 4,6-diamino-[1,7]naphthyridine-3-carbonitrile inhibitors of Tpl2 kinase and methods of making and using the same WYETH (US) 2008-10-07 US disclosed