SCHEMBL5141328

SCHEMBL5141328

CCOC(=O)c1cc(C#N)c(-n2ccc(CC(=O)NS(=O)(=O)Cc3ccccc3)c2)nc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 18/20 0.55
ALDH1A1 P00352 2/20 0.54
CHRM2 P08172 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133530 0.85 ALDH1A1 (0.58) P2RY12ALDH1A1
SCHEMBL3934625 0.80 ALDH1A1 (0.57) P2RY12ALDH1A1CHRM2CYP3A4CYP2C9
SCHEMBL3596659 0.80 P2RY12 (0.81) P2RY12ALDH1A1CHRM2CYP3A4CYP2C9
SCHEMBL3586432 0.80 P2RY12 (0.62) P2RY12ALDH1A1CHRM2CYP3A4CYP2C9
SCHEMBL3590489 0.79 P2RY12 (0.82) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3585028 0.75 P2RY12 (0.79) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3587890 0.74 P2RY12 (0.81) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3599495 0.74 P2RY12 (0.82) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3591594 0.74 P2RY12 (0.83) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3594087 0.73 P2RY12 (0.76) P2RY12CHRM2CYP3A4CYP2C9DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904474-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2008-04-02 EP disclosed
WO-2007008140-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2007-01-18 WO disclosed