SCHEMBL5141561

SCHEMBL5141561

N#CC(C(N)=O)c1ccc(F)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 3/20 0.42
APP P05067 1/20 0.40
CASP1 P29466 1/20 0.40
IDO1 P14902 1/20 0.39
S1PR3 Q99500 4/20 0.38
S1PR1 P21453 3/20 0.38
S1PR2 O95136 1/20 0.38
S1PR4 O95977 1/20 0.38
RAPGEF3 O95398 1/20 0.37
SLC2A1 P11166 1/20 0.36
RPA1 P27694 1/20 0.36
ICMT O60725 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802932 0.85 SLC6A3 (0.44) IDO1S1PR3S1PR1S1PR4TSHR
SCHEMBL4170313 0.84 MDM2 (0.42) MDM2S1PR3S1PR1S1PR2S1PR4
SCHEMBL1008191 0.82 MDM2 (0.40) MDM2S1PR3S1PR1S1PR2S1PR4
SCHEMBL6802464 0.80 HDAC4 (0.44) NPC1TSHR
SCHEMBL6802967 0.78 PARP1 (0.44) RAB9A
SCHEMBL12498059 0.77 MDM2 (0.46) MDM2APPCASP1IDO1S1PR3
SCHEMBL12497645 0.77 MDM2 (0.46) MDM2APPCASP1IDO1S1PR3
SCHEMBL21383218 0.76 LMNA (0.51) IDO1
SCHEMBL38655195 0.76 APP (0.64) MDM2APPCASP1IDO1ICMT
SCHEMBL5234318 0.76 APP (0.64) MDM2APPCASP1IDO1ICMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7297795-B2 Process for preparation of 4-amino-3-quinolinecarbonitriles WYETH HOLDINGS CORPORATION (US) 2007-11-20 US disclosed