SCHEMBL5144498

SCHEMBL5144498

CCCCN(Cc1ccc(OCc2ccccc2)cc1)Cc1c(-c2ccc(Cl)cc2)nc(-c2ccccc2)n1CCCC

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.46
MAPT P10636 1/20 0.45
ATP4A P20648 5/20 0.43
ATP4B P51164 5/20 0.43
RXFP1 Q9HBX9 1/20 0.41
DRD2 P14416 4/20 0.40
DRD3 P35462 4/20 0.40
HRH3 Q9Y5N1 1/20 0.40
C5AR1 P21730 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5072222 0.95 BCHE (0.50) BCHEATP4AATP4BDRD2DRD3
SCHEMBL5135937 0.94 ATP4A (0.49) MAPTATP4AATP4BRXFP1DRD2
SCHEMBL5135885 0.93 MAPT (0.45) MAPTATP4AATP4BRXFP1DRD2
SCHEMBL5136749 0.92 MAPT (0.48) MAPTATP4AATP4BRXFP1DRD2
SCHEMBL5136614 0.92 BCHE (0.49) BCHEATP4AATP4BDRD2DRD3
SCHEMBL5135970 0.91 BCHE (0.53) BCHEATP4AATP4BDRD2DRD3
SCHEMBL5134950 0.91 C5AR1 (0.45) BCHEMAPTATP4AATP4BC5AR1
SCHEMBL5135329 0.91 TP53 (0.46) BCHEMAPTATP4AATP4BDRD2
SCHEMBL5135824 0.90 C5AR1 (0.44) BCHEMAPTATP4AATP4BC5AR1
SCHEMBL5136524 0.90 C5AR1 (0.46) BCHEMAPTC5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed