SCHEMBL5072222

SCHEMBL5072222

CCCCN(Cc1ccc(OCc2ccccc2)cc1)Cc1c(-c2ccccc2)nc(-c2ccccc2)n1CCCC

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.50
ATP4A P20648 4/20 0.45
ATP4B P51164 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
C5AR1 P21730 1/20 0.42
MMP13 P45452 1/20 0.42
HRH3 Q9Y5N1 2/20 0.41
DRD2 P14416 4/20 0.41
DRD3 P35462 4/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5136614 0.97 BCHE (0.49) BCHEATP4AATP4BL3MBTL1C5AR1
SCHEMBL5135970 0.96 BCHE (0.53) BCHEATP4AATP4BL3MBTL1C5AR1
SCHEMBL5144498 0.95 BCHE (0.46) BCHEATP4AATP4BL3MBTL1C5AR1
SCHEMBL5070125 0.93 L3MBTL1 (0.51) BCHEATP4AATP4BL3MBTL1C5AR1
SCHEMBL5134960 0.93 ATP4A (0.52) ATP4AATP4BHRH3DRD2DRD3
SCHEMBL647665 0.92 ATP4A (0.46) ATP4AATP4BC5AR1HRH3DRD2
SCHEMBL5135786 0.92 BCHE (0.44) BCHEATP4AATP4BL3MBTL1C5AR1
SCHEMBL5137431 0.91 ATP4A (0.50) ATP4AATP4BHRH3DRD2DRD3
SCHEMBL5134735 0.90 ATP4A (0.51) ATP4AATP4BHRH3DRD2DRD3
SCHEMBL649161 0.90 C5AR1 (0.47) BCHEATP4AATP4BC5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed