SCHEMBL5145123

SCHEMBL5145123

CC(c1ccc(Cl)cc1)C(CNS(=O)(=O)c1cccc(Cl)c1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.53
MAPT P10636 6/20 0.50
KMT2A Q03164 6/20 0.50
MEN1 O00255 5/20 0.50
GAA P10253 5/20 0.50
TP53 P04637 4/20 0.50
THRB P10828 1/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
XBP1 P17861 1/20 0.47
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
PKM P14618 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5147475 0.96 PGR (0.56) PGRMAPTKMT2AMEN1GAA
SCHEMBL5146880 0.91 MAPT (0.59) MAPTKMT2AMEN1GAATP53
SCHEMBL5147423 0.90 KMT2A (0.56) MAPTKMT2AMEN1GAATP53
SCHEMBL5146669 0.89 MEN1 (0.60) MAPTKMT2AMEN1GAATP53
SCHEMBL5146784 0.86 CNR1 (0.65) CNR1CNR2
SCHEMBL5147326 0.85 MAPT (0.50) MAPTKMT2AMEN1GAATP53
SCHEMBL5147491 0.85 CA1 (0.51) PGRMAPTKMT2AMEN1GAA
SCHEMBL5145323 0.83 MEN1 (0.53) MAPTKMT2AMEN1GAATP53
SCHEMBL5145213 0.83 CA1 (0.54) MAPTKMT2AMEN1GAATP53
SCHEMBL5147402 0.83 CA1 (0.63) MAPTKMT2AMEN1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663113-A4 SUBSTITUTED SULFONAMIDES MERCK & CO INC (US) 2007-06-13 EP claimed
EP-1663113-A2 SUBSTITUTED SULFONAMIDES Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005027837-A2 SUBSTITUTED SULFONAMIDES MERCK & CO., INC. (US) 2005-03-31 WO claimed