SCHEMBL5147475

SCHEMBL5147475

CC(c1ccc(Cl)cc1)C(CNS(=O)(=O)c1cccc(Cl)c1)c1ccc(Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 7/20 0.56
KMT2A Q03164 3/20 0.48
GAA P10253 2/20 0.48
PKM P14618 2/20 0.48
ALDH1A1 P00352 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CNR2 P34972 2/20 0.46
CNR1 P21554 1/20 0.46
MAPT P10636 3/20 0.44
TP53 P04637 2/20 0.44
MEN1 O00255 2/20 0.44
HSD11B1 P28845 1/20 0.44
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
THRB P10828 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5145123 0.96 PGR (0.53) PGRKMT2AGAAPKMALDH1A1
SCHEMBL5147491 0.88 CA1 (0.51) PGRKMT2AGAAALDH1A1CA1
SCHEMBL5147423 0.88 KMT2A (0.56) KMT2AGAAPKMALDH1A1CA1
SCHEMBL5146784 0.87 CNR1 (0.65) CNR2CNR1
SCHEMBL5146880 0.87 MAPT (0.59) KMT2AGAAALDH1A1CA1CA2
SCHEMBL5147402 0.86 CA1 (0.63) KMT2AGAAALDH1A1CA1CA2
SCHEMBL5146645 0.85 CA1 (0.51) KMT2AGAAALDH1A1CA1CA2
SCHEMBL5146669 0.84 MEN1 (0.60) KMT2AGAAALDH1A1CA1CA2
SCHEMBL5145323 0.84 MEN1 (0.53) KMT2AGAAALDH1A1L3MBTL1CA1
SCHEMBL5147326 0.81 MAPT (0.50) KMT2AGAAALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663113-A4 SUBSTITUTED SULFONAMIDES MERCK & CO INC (US) 2007-06-13 EP claimed
EP-1663113-A2 SUBSTITUTED SULFONAMIDES Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005027837-A2 SUBSTITUTED SULFONAMIDES MERCK & CO., INC. (US) 2005-03-31 WO claimed