SCHEMBL5146760

SCHEMBL5146760

Cc1c(-c2cccnc2)[nH]c2cccc(CCCCCCCC(=O)O)c12

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 14/20 0.47
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
PARP1 P09874 1/20 0.41
MCL1 Q07820 1/20 0.38
FAAH O00519 1/20 0.38
CES1 P23141 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11167375 1.00 TBXAS1 (0.47) TBXAS1CYP11B1CYP11B2PARP1MCL1
SCHEMBL11172992 0.99 CYP11B1 (0.48) TBXAS1CYP11B1CYP11B2PARP1MCL1
SCHEMBL11167802 0.89 CYP11B1 (0.45) TBXAS1CYP11B1CYP11B2PARP1
SCHEMBL11164908 0.89 CYP11B1 (0.45) TBXAS1CYP11B1CYP11B2PARP1FAAH
SCHEMBL11167292 0.88 CYP11B1 (0.46) TBXAS1CYP11B1CYP11B2PARP1
SCHEMBL11174681 0.87 CYP11B1 (0.51) CYP11B1CYP11B2PARP1
SCHEMBL11164579 0.86 CYP11B1 (0.52) CYP11B1CYP11B2PARP1
SCHEMBL11162993 0.85 CYP11B1 (0.43) TBXAS1CYP11B1CYP11B2PARP1MCL1
SCHEMBL11175985 0.84 CYP11B1 (0.48) CYP11B1CYP11B2PARP1
SCHEMBL11168892 0.84 TBXAS1 (0.48) TBXAS1CYP11B1CYP11B2FAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242068-A4 ENDOGENOUS NITRIC OXIDE SYNTHESIS UNDER CONDITIONS OF LOW OXYGEN TENSION NITROMED INC (US) 2007-04-25 EP disclosed
EP-1242068-A1 ENDOGENOUS NITRIC OXIDE SYNTHESIS UNDER CONDITIONS OF LOW OXYGEN TENSION Nitromed, Inc. (US) 2002-09-25 EP disclosed
WO-2001089519-A1 THROMBOXANE INHIBITORS, COMPOSITIONS AND METHODS OF USE RELATED APPLICATIONS NITROMED, INC. (US) 2001-11-29 WO disclosed
WO-2001032167-A1 ENDOGENOUS NITRIC OXIDE SYNTHESIS UNDER CONDITIONS OF LOW OXYGEN TENSION NITROMED, INC. (US) 2001-05-10 WO disclosed
EP-0080154-A2 N-substituted 2-pyridyl indoles, process for their preparation, pharmaceutical compositions containing them, and their therapeutical use CIBA-GEIGY AG (CH) 1983-06-01 EP disclosed