SCHEMBL5146876

SCHEMBL5146876

CC(c1ccccc1)C(CNS(=O)(=O)C(C)(C)C)c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
MAPT P10636 4/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
LMNA P02545 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TP53 P04637 2/20 0.42
GAA P10253 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
XBP1 P17861 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ATM Q13315 1/20 0.41
CNR1 P21554 7/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5145543 1.00 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3MAPTMEN1
SCHEMBL5147333 0.95 CA1 (0.40) SLC6A2SLC6A4SLC6A3MAPTMEN1
SCHEMBL5145233 0.92 MAPT (0.37) SLC6A2SLC6A4SLC6A3MAPTKMT2A
SCHEMBL5147379 0.84 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3MAPTMEN1
SCHEMBL5143570 0.84 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3MAPTMEN1
SCHEMBL5146669 0.83 MEN1 (0.60) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL5146880 0.83 MAPT (0.59) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL5147423 0.81 KMT2A (0.56) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL5145330 0.80 CNR1 (0.46) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL5145391 0.79 CNR2 (0.36) CYP3A4CYP2C9CNR1CNR2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663113-A4 SUBSTITUTED SULFONAMIDES MERCK & CO INC (US) 2007-06-13 EP claimed
EP-1663113-A2 SUBSTITUTED SULFONAMIDES Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005027837-A2 SUBSTITUTED SULFONAMIDES MERCK & CO., INC. (US) 2005-03-31 WO claimed