SCHEMBL5147333

SCHEMBL5147333

CC(c1ccc(Cl)cc1)C(CNS(=O)(=O)C(C)(C)C)c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CNR1 P21554 5/20 0.39
GRIA4 P48058 2/20 0.36
CNR2 P34972 3/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
PTGES2 Q9H7Z7 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5145543 0.95 SLC6A2 (0.44) CA1CA2CNR1CNR2SLC6A2
SCHEMBL5146876 0.95 SLC6A2 (0.44) CA1CA2CNR1CNR2SLC6A2
SCHEMBL5145233 0.85 MAPT (0.37) GRIA4SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL5145391 0.84 CNR2 (0.36) CA1CA2CNR1GRIA4CNR2
SCHEMBL5147402 0.81 CA1 (0.63) CA1CA2MEN1KMT2AALDH1A1
SCHEMBL5147379 0.78 SLC6A2 (0.41) CA1CA2CNR1CNR2SLC6A2
SCHEMBL5143570 0.78 SLC6A2 (0.41) CA1CA2CNR1CNR2SLC6A2
SCHEMBL5147423 0.77 KMT2A (0.56) CA1CA2GRIA4MEN1KMT2A
SCHEMBL5147491 0.77 CA1 (0.51) CA1CA2CNR1CNR2MEN1
SCHEMBL5147331 0.77 RAB9A (0.43) CA1CA2CNR1CNR2PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663113-A4 SUBSTITUTED SULFONAMIDES MERCK & CO INC (US) 2007-06-13 EP claimed
EP-1663113-A2 SUBSTITUTED SULFONAMIDES Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005027837-A2 SUBSTITUTED SULFONAMIDES MERCK & CO., INC. (US) 2005-03-31 WO claimed