SCHEMBL5147205

SCHEMBL5147205

CC(C)(C)N1C[C@@H](O)C[C@H]1c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 12/20 0.55
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
CFB P00751 1/20 0.35
PIK3CD O00329 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22921054 1.00 RIPK1 (0.55) RIPK1MEN1KMT2APOLBHRH3
SCHEMBL22473311 0.83 RIPK1 (0.46) RIPK1MEN1KMT2APOLBHRH3
SCHEMBL30470257 0.82 RIPK1 (0.45) RIPK1HRH3
SCHEMBL454745 0.82 RIPK1 (0.46) RIPK1PIK3CD
SCHEMBL457570 0.82 RIPK1 (0.46) RIPK1PIK3CD
SCHEMBL454486 0.82 RIPK1 (0.46) RIPK1PIK3CD
SCHEMBL24774461 0.78 MEN1 (0.38) RIPK1MEN1KMT2ACHRNB4CHRNA3
SCHEMBL25587655 0.74 RIPK1 (0.53) RIPK1MEN1KMT2A
SCHEMBL30470290 0.73 RIPK1 (0.37) RIPK1MEN1KMT2APOLBHRH3
SCHEMBL22473213 0.72 RIPK1 (0.41) RIPK1CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551962-A4 MITOTIC KINESIN BINDING SITE MERCK & CO INC (US) 2007-08-01 EP disclosed
EP-1551962-A2 MITOTIC KINESIN BINDING SITE Merck & Co., Inc. (US) 2005-07-13 EP disclosed
WO-2004087050-A2 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2004-10-14 WO disclosed
WO-2004004652-A2 MITOTIC KINESIN BINDING SITE MERCK & CO., INC. (US) 2004-01-15 WO disclosed