SCHEMBL5147271

SCHEMBL5147271

O=C(Oc1cccc([N+](=O)[O-])c1CI)Oc1cccc([N+](=O)[O-])c1CI

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TDP1 Q9NUW8 4/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
RECQL P46063 1/20 0.44
HTT P42858 1/20 0.42
GPR35 Q9HC97 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 3/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
ESR2 Q92731 1/20 0.40
KCNH2 Q12809 1/20 0.39
APEX1 P27695 1/20 0.39
HSPB1 P04792 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148269 0.84 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL6513674 0.84 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL795687 0.81 KDM4E (0.43) ALDH1A1MEN1KMT2ATDP1RAB9A
SCHEMBL14642961 0.79 TDP1 (0.54) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL5047620 0.79 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ATDP1L3MBTL1
Bicarbonate SCHEMBL18955379 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2ATDP1L3MBTL1
Bicarbonate SCHEMBL18955378 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL57736 0.78 ALDH1A1 (0.60) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL29911025 0.78 ALDH1A1 (0.60) ALDH1A1MEN1KMT2ATDP1L3MBTL1
SCHEMBL3640407 0.77 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569895-A4 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT INC (US) 2007-07-11 EP disclosed
EP-1569895-A1 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF Xenoport, Inc. (US) 2005-09-07 EP disclosed
EP-1404324-A4 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT INC (US) 2004-12-22 EP disclosed
WO-2004052844-A1 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT, INC. (US) 2004-06-24 WO disclosed
EP-1404324-A2 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF Xenoport, Inc. (US) 2004-04-07 EP disclosed
WO-2002100347-A2 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT, INC. (US) 2002-12-19 WO disclosed