SCHEMBL5147300

SCHEMBL5147300

CC(NS(=O)(=O)c1cccc(-c2ccccc2)c1)C(Cc1ccc(Cl)cc1)Oc1ccc(Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.59
CNR2 P34972 7/20 0.59
ADAMTS5 Q9UNA0 1/20 0.46
MMP2 P08253 1/20 0.46
PPARG P37231 2/20 0.46
PPARA Q07869 2/20 0.46
CTSL P07711 5/20 0.44
CTSS P25774 5/20 0.44
CTSB P07858 4/20 0.44
CTSK P43235 4/20 0.44
ADAMTS4 O75173 1/20 0.42
MMP13 P45452 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5585077 0.90 CNR1 (0.53) CNR1CNR2ADAMTS5MMP2PPARG
SCHEMBL14512665 0.89 CNR1 (0.48) CNR1CNR2PPARGPPARAADAMTS4
SCHEMBL5585088 0.88 CNR1 (0.53) CNR1CNR2ADAMTS5MMP2PPARG
SCHEMBL5177950 0.85 CNR1 (0.48) CNR1CNR2ADAMTS5MMP2PPARG
SCHEMBL5145056 0.83 CNR1 (0.53) CNR1CNR2PPARGPPARA
SCHEMBL5142976 0.82 CNR1 (0.61) CNR1CNR2ADAMTS4MMP13
SCHEMBL5145180 0.81 CNR1 (0.47) CNR1CNR2ADAMTS5MMP2
SCHEMBL5584867 0.78 CNR1 (0.50) CNR1CNR2ADAMTS5MMP2
SCHEMBL5145119 0.73 CNR1 (0.76) CNR1CNR2
SCHEMBL5146878 0.70 CNR1 (0.74) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663113-A4 SUBSTITUTED SULFONAMIDES MERCK & CO INC (US) 2007-06-13 EP claimed
US-20070105914-A1 Substituted sulfonamides MERCK SHARP & DOHME CORP. 2007-05-10 US claimed
EP-1663113-A2 SUBSTITUTED SULFONAMIDES Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005027837-A2 SUBSTITUTED SULFONAMIDES MERCK & CO., INC. (US) 2005-03-31 WO claimed
US-20070105914-A1 Substituted sulfonamides MERCK SHARP & DOHME CORP. 2007-05-10 US disclosed
US-20070105914-A1 Substituted sulfonamides MERCK SHARP & DOHME CORP. 2007-05-10 US disclosed
US-20070105914-A1 Substituted sulfonamides MERCK SHARP & DOHME CORP. 2007-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070105914-A1 Substituted sulfonamides CNR2, CNR1, FAAH CNR1 2/4885CNR2 1/4885ADAMTS5 827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.